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Lisinopril: uses, Dosage, Side Effects, indications

Look for Drugs and Conditions

Lisinopril

Lisinopril

Inhibition of ACE by lisinopril reduces the plasma angiotensin II levels which lead to vasodilation and reduction of aldosterone secretion thus lowering the blood pressure.

Indications

All grades of hypertension, hypertension complicated by diabetes mellitus, gout, asthma & mental depression. Congestive cardiac failure.


Dosage

Hypertension; Initially 10 mg once daily Maint. dose 20-40 mg/day. Max. 80 mg once daily. C.C.F.; Initially 2.5 mg once daily. Maint dose 5-20 mg once daily.


Contra-Indications

Hypersensitivity, aortic stenosis, outflow obstruction, angioedema related to previous treatment with ACE inhibitor, pregnancy, children, nursing mothers.


Special Precautions

Renal impairment, lisinopril may cause hypotension in patients undergoing major surgery or during anaesthesia. In severe C.C.F. it may cause oliguria and/or progressive azotemia & rarely acute renal failure. Paediatrics: Contraindicated. Pregnancy: Contraindicated. Lactation: Drug passes into breast milk hence containdicated. Elderly: Reduced dose may be necessary.


Side Effects

Headache, dizziness, cough, hyper-kalaemia, diarrhoea, angioedema, hypotension.


Drug Interactions

Indomethacin may reduce hypotensive effect. Hydrochlorothiazide may potentiate antihypertensive effect. Raised serum lithium levels, hypotensive effect potentiated by alcohol. Inhibit tachycardia produced by vasodialators. Co-administration of cyclo-oxy-genase inhibitors cause reducton in renal function.


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