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Fondaparinux Sodium- Dosage, Side Effects, indications, Uses and Precaution

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Fondaparinux Sodium

Fondaparinux Sodium

it is an anticoagulant medication chemically related to low molecular weight heparins. The antithrombotic activity of fondaparinux is the result of ATIII-mediated selective inhibition of Factor Xa. By selectively binding to ATIII, Fondaparinux potentiates (about 300 times) the neutralization of Factor Xa by ATIII. Neutralization of Factor Xa interrupts the blood coagulation cascade and thus inhibits thrombin formation and thrombus development. It is thought that fondaparinux is unlikely to induce thrombocytopenia via a heparin-induced thrombocytopenia (HIT)-like mechanism given its chemical structure. As a result, fondaparinux has been used as an alternative anticoagulant in heparin-induced thrombocytopenia (HIT) patients.

Indications

prophylaxis of deep vein thrombosis (DVT), which may lead to pulmonary embolism (PE): • In patients undergoing hip fracture surgery, including extended prophylaxis; • In patients undergoing hip replacement surgery; • In patients undergoing knee replacement surgery; • In patients undergoing abdominal surgery who are at risk for thromboembolic complications. For treatment of acute pulmonary embolism


Dosage

SC; 25 mg


Contra-Indications

Severe renal impairment • Active major bleeding. • Bacterial endocarditis. • Thrombocytopenia associated with a positive in vitro test for anti-platelet antibody in the presence of fondaparinux sodium. • Body weight


Special Precautions

Paediatrics: Safety not yet established Pregnancy: Category B, use if needed Lactation: Not known if excreted in milk Elderly: Risk of side effects increases with age


Side Effects

Anaemia, bleeding, purpura, oedema.


Other Brands With Same Generic
Brand Name Manufactured by
ARIXTRA GSK

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